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MCE 國際站:Ionomycin calcium
品牌:MedChemExpress (MCE)
CAS:56092-82-1
純度:≥98.0%
貨號:HY-13434A
中文名稱:離子霉素鈣鹽
Synonyms:SQ23377 calcium
存儲條件:4°C,密封保存,遠(yuǎn)離潮濕 *溶劑中:-80°C,6個(gè)月;-20°C,1個(gè)月(密封保存,遠(yuǎn)離潮濕)
運(yùn)輸條件:美國大陸的室溫;其他地方可能有所不同。
產(chǎn)品活性:Ionomycin calcium (SQ23377 calcium) 是一種有效的,選擇性的鈣離子載體 (calcium ionophore),也是一種由 Streptomyces conglobatus 產(chǎn)生的抗生素。Ionomycin calcium (SQ23377 calcium) 對二價(jià)陽離子具有高度特異性 (Ca>Mg>Sr=Ba)。Ionomycin (SQ23377) 促進(jìn)細(xì)胞凋亡。Ionomycin calcium (SQ23377 calcium) 還誘導(dǎo)蛋白激酶C (PKC) 激活。
IC50 & Target:Calcium ionophore[1]
熱銷產(chǎn)品:Masitinib | Potassium 1H-indol-3-yl sulfate | Ouabain (Octahydrate) | L-778123 (hydrochloride) | Romosozumab | CHAPS | 1,2-Distearoyl-sn-glycero-3-phosphorylcholine | Denosumab | Cobimetinib | N,N,N′,N′-Tetracyclohexyl-3-oxapentanediamide
Trending products:Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | Isotope-Labeled Compounds | Oligonucleotides
參考文獻(xiàn):
[1]. Liu C,et al. Characterization of ionomycin as a calcium ionophore. J Biol Chem. 1978 Sep 10;253(17):5892-4.
[2]. Chatila T, et al. Mechanisms of T cell activation by the calcium ionophore ionomycin. J Immunol. 1989 Aug 15;143(4):1283-9.
[3]. Gil-Parrado S, et al. Ionomycin-activated calpain triggers apoptosis. A probable role for Bcl-2 family members. J Biol Chem. 2002 Jul 26;277(30):27217-26.
[4]. Stoeck A, et al A role for exosomes in the constitutive and stimulus-induced ectodomain cleavage of L1 and CD44. Biochem J. 2006 Feb 1;393(Pt 3):609-18.
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